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SYS · ONLINEPASS · 63.0%
Open Assay
Independent Testing / Est. 2026
BATCH04·26·B
PASS63.0%
N27
§ 01 / Reference

Peptide index

209 compounds catalogued. Each entry is graded on evidence strength. Blind-purchase testing data appears as the independent assay program comes online.

209
Compounds
49
Tier 1
63
Speculative
Mean pass
Search
Evidence tier
Category
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209 / 209
#Compound Also known asCategory Evidence Pass % N Supp.
015-Amino 1MQ
Small-molecule nicotinamide N-methyltransferase (NNMT) inhibitor (not a peptide; commonly sold in peptide-market channels)
OtherSPECULATIVE
025-Amino-1MQ + NADH (Blend)
Two-component blend - 5-Amino-1-methylquinolinium (5-A1MQ; selective NNMT inhibitor small molecule) + NADH (reduced nicotinamide adenine dinucleotide)
MetabolicTIER 3 · Preclinical
039-Me-BC
β-carboline alkaloid (small molecule); proposed dopamine system upregulator
CognitiveSPECULATIVE
04Ac2-26
Synthetic N-acetylated 25-residue peptide derived from Annexin A1 N-terminus
Healing, ImmuneTIER 3 · Preclinical
05ACE-031
Recombinant human activin receptor type IIB extracellular domain — IgG1 Fc fusion protein
GH-stackTIER 2 · Translational
06Acetyl Hexapeptide-8
Synthetic N-acetylated hexapeptide; INCI 'Acetyl Hexapeptide-8'; SNAP-25 mimic / SNARE-targeting cosmetic peptide
CosmeticSPECULATIVE
07Acetyl Tetrapeptide-11
Synthetic acetylated tetrapeptide; INCI 'Acetyl Tetrapeptide-11'; tenascin-X / dermal density cosmetic peptide
CosmeticSPECULATIVE
08Acetyl Tetrapeptide-2
Synthetic acetylated tetrapeptide; INCI 'Acetyl Tetrapeptide-2'; thymus-derived cosmetic peptide
CosmeticSPECULATIVE
09Acetyl Tetrapeptide-5
Synthetic acetylated tetrapeptide; INCI 'Acetyl Tetrapeptide-5'; periorbital edema / under-eye cosmetic peptide
CosmeticSPECULATIVE
10Acetyl Tetrapeptide-9
Synthetic acetylated tetrapeptide; INCI 'Acetyl Tetrapeptide-9'; dermal density cosmetic peptide
CosmeticSPECULATIVE
11ACTH 1-24
Synthetic 24-residue N-terminal fragment of ACTH (corticotropin); MC2R agonist
Cognitive, ImmuneTIER 1 · Clinical
12Adrafinil
Pro-drug of modafinil (small molecule, hydroxyamide of modafinil)
CognitiveTIER 2 · Translational
13AHK-Cu
Copper-binding tripeptide; alanyl-histidyl-lysine copper complex (analog of GHK-Cu)
CosmeticTIER 3 · Preclinical
14AICAR
Synthetic AMP-mimetic small molecule; AMPK activator (acadesine)
MetabolicTIER 2 · Translational
15Albiglutide
Recombinant GLP-1-(7-37) fusion to human serum albumin (long-acting GLP-1 receptor agonist)
MetabolicTIER 1 · Clinical
16Alpha-GPC
Cholinergic precursor (small molecule, glycerylphosphorylcholine)
CognitiveTIER 2 · Translational
17Amylin (native)
Endogenous 37-residue islet amyloid polypeptide; co-secreted with insulin from beta-cells; CTR/RAMP-amylin receptor agonist
MetabolicTIER 3 · Preclinical
18Anamorelin
Non-peptide ghrelin receptor (GHS-R1a) agonist (small molecule)
GH secretagogue, MetabolicTIER 2 · Translational
19ANP-28 (Atrial Natriuretic Peptide)
Endogenous 28-residue atrial natriuretic peptide; NPR-A receptor agonist
MetabolicTIER 3 · Preclinical
20AOD-9604
Modified fragment of human growth hormone amino acids 176-191
MetabolicTIER 3 · Preclinical
21ARA-290
11-amino-acid peptide derived from erythropoietin; innate repair receptor (IRR) agonist
HealingTIER 2 · Translational
22B7-33
Modified single-chain relaxin-2 analog; biased RXFP1 receptor agonist
HealingSPECULATIVE
23BAM-15
Selective mitochondrial protonophore uncoupler (small molecule)
Metabolic, LongevityTIER 3 · Preclinical
24BDNF (Brain-Derived Neurotrophic Factor)
Endogenous neurotrophin (TrkB receptor ligand); recombinant
CognitiveTIER 3 · Preclinical
25BMP-7
Recombinant human bone morphogenetic protein (TGF-β superfamily ligand)
HealingTIER 1 · Clinical
26BNP-32 (B-type Natriuretic Peptide)
Endogenous 32-residue B-type natriuretic peptide; NPR-A agonist; ventricular myocyte source
MetabolicTIER 1 · Clinical
27BPC-157
Synthetic 15-amino-acid pentadecapeptide
HealingTIER 3 · Preclinical
28BPC-157 + TB-500 (Wolverine Blend)
Multi-component research-peptide blend
Blend, HealingTIER 3 · Preclinical
29Bremelanotide
Synthetic cyclic heptapeptide analog of alpha-MSH; non-selective melanocortin receptor agonist
OtherTIER 1 · Clinical
30Bronchogen
Khavinson-tradition tetrapeptide (Ala-Glu-Asp-Leu); proposed bronchial epithelium bioregulator
Longevity, ImmuneSPECULATIVE
31Cagrilintide
Long-acting amylin analog; AMY1/2/3 receptor agonist
MetabolicTIER 2 · Translational
32CagriSema
Fixed-ratio coformulation: cagrilintide (amylin agonist) plus semaglutide (GLP-1 agonist)
MetabolicTIER 2 · Translational
33Calcitonin
32-amino-acid peptide hormone; calcitonin receptor agonist; salmon-derived form is most clinically used
OtherTIER 1 · Clinical
34Calcitonin (salmon)
Synthetic salmon calcitonin analog (32-residue peptide)
MetabolicTIER 1 · Clinical
35Calcitonin Gene-Related Peptide (CGRP)
Endogenous 37-residue calcitonin gene-related peptide; CGRP receptor (CALCRL/RAMP1) agonist
CognitiveTIER 1 · Clinical
36Capromorelin
Non-peptide ghrelin receptor (GHS-R1a) agonist (spiroindoline class)
GH secretagogueTIER 1 · Clinical
37Cardiogen
Khavinson-tradition tripeptide (Ala-Glu-Asp); proposed cardiac muscle bioregulator
LongevitySPECULATIVE
38Cartalax
Khavinson-tradition tripeptide; proposed cartilage bioregulator
Longevity, HealingSPECULATIVE
39Cerebrolysin
Porcine-brain-derived peptide preparation (low-molecular-weight neuropeptides plus free amino acids)
CognitiveTIER 2 · Translational
40Chelohart
Khavinson-tradition cardiac muscle bioregulator (variant)
LongevitySPECULATIVE
41Chitomur
Khavinson-tradition urinary bladder muscle bioregulator (KE-class)
LongevitySPECULATIVE
42Cholecystokinin-33
Endogenous 33-residue gut peptide; CCK-A and CCK-B receptor agonist; full-length form (the 8mer sincalide is the synthetic clinical analog)
Cognitive, MetabolicTIER 3 · Preclinical
43Chonluten
Khavinson-tradition tripeptide (Glu-Asp-Gly); proposed chondrogenic / bronchopulmonary bioregulator
LongevitySPECULATIVE
44Citicoline
CDP-choline (small molecule, nucleotide-choline conjugate)
CognitiveTIER 2 · Translational
45CJC-1295
Tetrasubstituted GHRH(1-29) analog; DAC variant covalently binds albumin for extended half-life
GH secretagogueSPECULATIVE
46CJC-1295 + Ipamorelin (Blend)
Two-component vendor blend — CJC-1295 (with or without DAC; vendors vary) plus ipamorelin (selective GHS-R1a hexapeptide)
Blend, GH-stackSPECULATIVE
47CJC-1295 with DAC
Modified human GHRH(1-29) analog with drug-affinity-complex (DAC) maleimide group for covalent albumin binding
GH secretagogueSPECULATIVE
48CJC-1295 without DAC
Tetrasubstituted human GHRH(1-29) analog (D-Ala2, Gln8, Ala15, Leu27)
GH secretagogueSPECULATIVE
49Coenzyme Q10 (injectable)
Coenzyme Q10 (ubiquinone); injectable research-grade preparation; mitochondrial electron transport cofactor
Longevity, MetabolicTIER 2 · Translational
50Cortagen
Khavinson-tradition tetrapeptide (Ala-Glu-Asp-Pro); proposed cerebral cortex bioregulator
Longevity, CognitiveSPECULATIVE
51Cortistatin
Endogenous somatostatin-family neuropeptide; binds somatostatin receptors SSTR1 through SSTR5 with comparable affinity to somatostatin, plus the ghrelin receptor (GHS-R1a) and (in mast cells) MrgX2 — a broader receptor profile than somatostatin
Cognitive, ImmuneTIER 3 · Preclinical
52Crystagen
Khavinson-tradition tripeptide (Glu-Asp-Pro); proposed immune bioregulator
Longevity, ImmuneSPECULATIVE
53Danuglipron
Oral small-molecule GLP-1 receptor agonist (Pfizer)
MetabolicTIER 2 · Translational
54Dermorphin
7-amino-acid peptide (Tyr-D-Ala-Phe-Gly-Tyr-Pro-Ser-NH2) from amphibian skin; mu-opioid agonist
OtherSPECULATIVE
55Desmopressin
Synthetic analog of vasopressin; selective V2-receptor agonist
OtherTIER 1 · Clinical
56Dihexa
Synthetic hexapeptide; angiotensin IV analog
CognitiveSPECULATIVE
57Dipeptide Diaminobutyroyl Benzylamide Diacetate
Synthetic snake-venom mimetic dipeptide; Waglerin-1-derived; nicotinic acetylcholine receptor antagonist; INCI 'Dipeptide Diaminobutyroyl Benzylamide Diacetate'
CosmeticSPECULATIVE
58DSIP
9-amino-acid peptide isolated from rabbit brain in 1977
CognitiveTIER 3 · Preclinical
59Dulaglutide
GLP-1 analog fused to IgG4 Fc fragment; long-acting GLP-1 receptor agonist
MetabolicTIER 1 · Clinical
60Dutasteride
Dual 5-alpha-reductase inhibitor (type 1 and type 2; small molecule)
CosmeticTIER 1 · Clinical
61Ecnoglutide
Biased GLP-1 receptor agonist (functional selectivity for cAMP over beta-arrestin)
MetabolicTIER 2 · Translational
62Efpeglenatide
Long-acting GLP-1 receptor agonist with glucagon receptor selectivity (Hanmi/Sanofi)
MetabolicTIER 2 · Translational
63EGF (Epidermal Growth Factor)
Recombinant human epidermal growth factor; EGFR ligand
Cosmetic, HealingTIER 2 · Translational
64Enclomiphene
Selective estrogen receptor modulator (SERM); trans-isomer of clomiphene citrate
Sexual / hormonalTIER 2 · Translational
65Endoluten
Khavinson-tradition extended pineal bioregulator (AEDG-related; epitalon analog)
LongevitySPECULATIVE
66Epitalon
Synthetic tetrapeptide Ala-Glu-Asp-Gly
CognitiveSPECULATIVE
67Exenatide
Synthetic version of exendin-4 (Gila monster saliva); GLP-1 receptor agonist
MetabolicTIER 1 · Clinical
68Fasoracetam
Racetam-class nootropic (small molecule); proposed mGluR3 / Group II metabotropic glutamate receptor agonist
CognitiveTIER 2 · Translational
69FGF-2 (Basic Fibroblast Growth Factor)
Recombinant basic fibroblast growth factor; FGFR1c agonist (and FGFR2/3/4 binding)
Cosmetic, HealingTIER 2 · Translational
70FGF-21 (Fibroblast Growth Factor 21)
Endogenous fibroblast growth factor 21; beta-Klotho/FGFR1c receptor complex agonist
Metabolic, LongevityTIER 2 · Translational
71Finasteride
Selective 5-alpha-reductase type 2 inhibitor (small molecule)
CosmeticTIER 1 · Clinical
72Follistatin + B-Complex (SlimAssist Blend)
Two-component blend — recombinant follistatin (FST-315 or FST-344, vendor-dependent) plus B-vitamin complex (composition varies)
Blend, GH-stackSPECULATIVE
73Follistatin-315 (FST-315)
Native follistatin short isoform (315 residues; predominant circulating form)
GH-stackTIER 3 · Preclinical
74Follistatin-344 (FST-344)
Native follistatin long isoform (344 residues; high heparan sulfate binding, tissue-retained)
GH-stackTIER 3 · Preclinical
75FOXO4-DRI
D-amino-acid retro-inverso peptide designed to interfere with FOXO4-p53 interaction
CognitiveSPECULATIVE
76GDNF (Glial Cell Line-Derived Neurotrophic Factor)
Endogenous neurotrophin (TGF-beta superfamily; RET receptor signalling); recombinant
CognitiveTIER 2 · Translational
77GHK (Glycyl-Histidyl-Lysine)
Native tripeptide glycyl-histidyl-lysine (GHL); copper-free form
Cosmetic, HealingTIER 3 · Preclinical
78GHK-Cu
Naturally occurring tripeptide (Gly-His-Lys) complexed with copper(II)
HealingTIER 2 · Translational
79Ghrelin (native)
Endogenous 28-residue peptide hormone (octanoylated at Ser3) — primary GHS-R1a ligand
GH secretagogue, MetabolicTIER 3 · Preclinical
80GHRP-2
Synthetic hexapeptide; ghrelin / GHS-R1a receptor agonist
GH secretagogueTIER 2 · Translational
81GHRP-6
Synthetic hexapeptide; ghrelin / GHS-R1a receptor agonist; first characterized GHRP
GH secretagogueSPECULATIVE
82GHRP-7
Synthetic hexapeptide growth-hormone-releasing peptide (GHS-R1a agonist class)
GH secretagogueSPECULATIVE
83Glandokort
Khavinson-tradition adrenal cortex bioregulator
LongevitySPECULATIVE
84GLP-2 (native)
Endogenous 33-residue intestinotrophic gut peptide; cleaved from proglucagon
MetabolicTIER 1 · Clinical
85Glucagon (rescue)
Recombinant 29-residue glucagon peptide; native glucagon receptor agonist
MetabolicTIER 1 · Clinical
86Glucagon-like Peptide-1 (native)
Endogenous 30- or 31-residue intestinotrophic gut peptide (GLP-1(7-36)NH2 or GLP-1(7-37)); GLP-1R agonist
MetabolicTIER 1 · Clinical
87Glutathione
Tripeptide; endogenous antioxidant (not a classical peptide hormone)
OtherTIER 2 · Translational
88Glycine (research-grade spray)
Endogenous non-essential amino acid; NMDA glycine-binding site agonist
Longevity, CognitiveTIER 2 · Translational
89Gonadorelin
Native human gonadotropin-releasing hormone — decapeptide
Sexual / hormonalTIER 1 · Clinical
90HCG (Human Chorionic Gonadotropin)
Glycoprotein heterodimer — α-subunit (common to LH, FSH, TSH) plus hCG-specific β-subunit
Sexual / hormonalTIER 1 · Clinical
91Hexapeptide-11
Synthetic hexapeptide; INCI 'Hexapeptide-11'; anti-senescence cosmetic peptide
Cosmetic, LongevitySPECULATIVE
92Hexapeptide-40
Synthetic hexapeptide; INCI 'Hexapeptide-40'; sirtuin-1 (SIRT1) activating cosmetic peptide
Cosmetic, LongevitySPECULATIVE
93Hexapeptide-44
Synthetic hexapeptide; INCI 'Hexapeptide-44'; lamin B1 upregulating cosmetic peptide
Cosmetic, LongevitySPECULATIVE
94Hexarelin
Synthetic hexapeptide; potent ghrelin/GHS-R1a agonist; also CD36 ligand
GH secretagogueTIER 3 · Preclinical
95HGH Fragment 176-191 (AOD-9604)
Synthetic 16-residue C-terminal fragment of human growth hormone (residues 176-191); proposed lipolytic without GH-axis activation
MetabolicTIER 2 · Translational
96Honluten
Khavinson-tradition tripeptide (Lys-Glu-Asp); proposed lung tissue bioregulator
LongevitySPECULATIVE
97Humanin
24-amino-acid mitochondrial-derived peptide encoded within the MT-RNR2 gene
CognitiveTIER 3 · Preclinical
98IGF-1 LR3
Modified IGF-1 analog with N-terminal extension and Arg-for-Glu substitution at position 3; reduced IGFBP affinity
GH secretagogueSPECULATIVE
99Insulin and insulin analogs
Class page — recombinant human insulin and engineered analogs (rapid: lispro, aspart, glulisine; long: glargine, detemir, degludec; ultra-long: icodec)
MetabolicTIER 1 · Clinical
100Ipamorelin
Pentapeptide (Aib-His-D-2-Nal-D-Phe-Lys-NH2) ghrelin / GHS-R1a receptor agonist
GH secretagogueSPECULATIVE
101Kisspeptin-10
10-amino-acid C-terminal fragment of kisspeptin; KISS1R (GPR54) receptor agonist
OtherTIER 2 · Translational
102KPV (Lys-Pro-Val)
Synthetic tripeptide — C-terminal fragment of α-MSH (residues 11-13)
Healing, ImmuneTIER 3 · Preclinical
103L-Carnitine
Endogenous quaternary ammonium small molecule; mitochondrial fatty-acid transporter cofactor
MetabolicTIER 2 · Translational
104Leuprolide
Synthetic GnRH (gonadotropin-releasing hormone) superagonist — nonapeptide-amide
Sexual / hormonalTIER 1 · Clinical
105Liquid Glutathione
Reduced glutathione (GSH); endogenous tripeptide antioxidant (gamma-Glu-Cys-Gly)
LongevityTIER 2 · Translational
106Liraglutide
Acylated GLP-1 receptor agonist; predecessor of semaglutide
MetabolicTIER 1 · Clinical
107Livagen
Khavinson-tradition tetrapeptide (Lys-Glu-Asp-Ala); proposed liver bioregulator
LongevitySPECULATIVE
108Lixisenatide
Synthetic 44-residue exendin-4 analog; short-acting GLP-1 receptor agonist
MetabolicTIER 1 · Clinical
109LL-37
37-amino-acid cationic antimicrobial peptide; human cathelicidin
HealingTIER 3 · Preclinical
110Maralixibat
Selective ileal bile acid transporter (IBAT/ASBT) inhibitor (small molecule)
MetabolicTIER 1 · Clinical
111Matrixyl
Synthetic palmitoylated pentapeptide; INCI 'Palmitoyl Pentapeptide-4'; collagen-stimulating cosmetic peptide
CosmeticSPECULATIVE
112Mazdutide
Dual GLP-1 / glucagon receptor agonist (Innovent Biologics + Eli Lilly co-development)
MetabolicTIER 2 · Translational
113Melanotan II
Synthetic cyclic heptapeptide analog of alpha-MSH; broad melanocortin receptor agonist
OtherTIER 3 · Preclinical
114Melanotan-1 (Afamelanotide)
Synthetic alpha-MSH analog; cyclic 13-residue peptide; MC1R-selective melanocortin agonist
Cosmetic, Sexual / hormonalTIER 1 · Clinical
115Metformin
Biguanide-class oral antihyperglycaemic (small molecule); complex I inhibition; AMPK activator
Longevity, MetabolicTIER 1 · Clinical
116Methylene Blue
Phenothiazine dye (small molecule); mitochondrial alternative electron carrier; MAO inhibitor at high doses
Longevity, CognitiveTIER 1 · Clinical
117MGF
Synthetic peptide — C-terminal E-domain of the IGF-1Ec splice variant
GH-stackTIER 3 · Preclinical
118Minoxidil
Vasodilator small molecule; ATP-sensitive potassium channel opener
CosmeticTIER 1 · Clinical
119MK-677
Non-peptide spiroindoline small molecule; oral ghrelin / GHS-R1a receptor agonist
GH secretagogueTIER 2 · Translational
120Modafinil
Wakefulness-promoting agent (small molecule, sulfinyl class)
CognitiveTIER 1 · Clinical
121Motilin
Endogenous 22-residue gut peptide; motilin receptor (MLNR/GPR38) agonist
CognitiveTIER 3 · Preclinical
122MOTS-c
16-amino-acid mitochondrial-derived peptide encoded within the 12S rRNA gene
MetabolicTIER 3 · Preclinical
123Myostatin Inhibitor (research class)
Heterogeneous class — soluble receptor decoys (ACE-031), monoclonal antibodies (domagrozumab, taldefgrobep), engineered peptide ligands. Vendor product chemistry is typically unspecified.
GH-stackTIER 3 · Preclinical
124Myristoyl Pentapeptide-17
Synthetic myristoylated pentapeptide; INCI 'Myristoyl Pentapeptide-17'; eyelash growth cosmetic peptide
CosmeticSPECULATIVE
125N-Acetyl-Selank
N-acetylated heptapeptide; Russian-origin nootropic; modified Selank for stability
CognitiveSPECULATIVE
126N-Acetyl-Semax-Amidate
Modified heptapeptide derivative of Semax (ACTH(4-10) analog); N-acetylated and C-amidated for stability
CognitiveSPECULATIVE
127NAD
Endogenous nicotinamide adenine dinucleotide; NAD+ research compound (injectable / IV)
LongevityTIER 2 · Translational
128Nesiritide
Recombinant 32-residue B-type natriuretic peptide (BNP-32); NPR-A receptor agonist
MetabolicTIER 1 · Clinical
129Neuropeptide Y
Endogenous 36-residue hypothalamic neuropeptide; pancreatic polypeptide family; Y1-Y5 receptor agonist
CognitiveTIER 3 · Preclinical
130NGF (Nerve Growth Factor)
Endogenous neurotrophin (beta-subunit homodimer of NGF complex); recombinant
CognitiveTIER 2 · Translational
131NMN
Nicotinamide mononucleotide; NAD+ precursor (small molecule)
LongevityTIER 2 · Translational
132Noopept
Synthetic peptide-derived nootropic (small molecule); cleaves to bioactive cyclic prolyl-glycine in vivo
CognitiveTIER 3 · Preclinical
133NR
Nicotinamide riboside; NAD+ precursor (small molecule)
LongevityTIER 2 · Translational
134Octreotide
Synthetic cyclic octapeptide analog of somatostatin; SSTR2/SSTR5 agonist
OtherTIER 1 · Clinical
135Orforglipron
Oral small-molecule GLP-1 receptor agonist (Eli Lilly, biased)
MetabolicTIER 2 · Translational
136Osteogenic Peptide (BMP-mimetic class)
Heterogeneous class — synthetic peptides typically 15-30 residues derived from BMP-2 or BMP-7 knuckle-epitope regions
HealingTIER 3 · Preclinical
137Ovagen
Khavinson-tradition liver/ovarian bioregulator (Glu-Asp-Leu and related)
LongevitySPECULATIVE
138Oxyntomodulin
Endogenous 37-residue dual GLP-1 + glucagon receptor agonist; cleavage product of proglucagon
MetabolicTIER 3 · Preclinical
139Oxytocin
Nonapeptide (9 amino acids with disulfide bond); OT receptor agonist
OtherTIER 1 · Clinical
140P-21
Synthetic 11-residue peptide derived from a region of ciliary neurotrophic factor (CNTF); proposed neurogenic and neuroprotective agent
CognitiveTIER 3 · Preclinical
141Palmitoyl Hexapeptide-12
Synthetic palmitoylated hexapeptide; INCI 'Palmitoyl Hexapeptide-12'; elastin-stimulating cosmetic peptide
CosmeticSPECULATIVE
142Palmitoyl Tetrapeptide-7
Synthetic palmitoylated tetrapeptide; INCI 'Palmitoyl Tetrapeptide-7'; anti-inflammatory cosmetic peptide
CosmeticSPECULATIVE
143Palmitoyl Tripeptide-1
Synthetic palmitoylated tripeptide; INCI 'Palmitoyl Tripeptide-1'; topicalised GHK (palmitoyl-glycyl-histidyl-lysine)
CosmeticSPECULATIVE
144Palmitoyl Tripeptide-5
Synthetic palmitoylated tripeptide; INCI 'Palmitoyl Tripeptide-5'; TGF-β mimetic cosmetic peptide
CosmeticSPECULATIVE
145Pancragen
Khavinson-tradition tetrapeptide (Lys-Glu-Asp-Trp); proposed pancreatic islet bioregulator
LongevitySPECULATIVE
146Pasireotide
Multireceptor somatostatin analog; cyclohexapeptide; binds SSTR1, SSTR2, SSTR3, and SSTR5 with high affinity (broader profile than octreotide which is selective for SSTR2)
Cognitive, MetabolicTIER 1 · Clinical
147PDA (Pentadeca-Arginate)
Arginate salt formulation of the BPC-157 pentadecapeptide sequence
HealingTIER 3 · Preclinical
148PDRN (Polydeoxyribonucleotide)
Polydeoxyribonucleotide; salmon-DNA fragments (50 to 1500 base pairs typical); A2A adenosine receptor agonist
Cosmetic, HealingTIER 2 · Translational
149PE 22-28
7-amino-acid fragment of B-cell-derived PEPITEM protein
HealingSPECULATIVE
150PEG-MGF
PEGylated synthetic peptide (MGF E-domain 24mer with PEG conjugation; PEG MW unspecified by vendors)
GH-stackTIER 3 · Preclinical
151Pentapeptide-3
Synthetic pentapeptide; INCI 'Pentapeptide-3'; nicotinic acetylcholine receptor blocker (topical)
CosmeticSPECULATIVE
152Peptide YY (PYY)
Endogenous 36-residue peptide YY; pancreatic polypeptide family; Y2 receptor preferred (especially PYY 3-36)
MetabolicTIER 3 · Preclinical
153Phenibut
GABA-B receptor agonist (small molecule, β-aryl-GABA derivative)
CognitiveTIER 2 · Translational
154Pinealon
Synthetic tetrapeptide; Khavinson-tradition pineal bioregulator; sequence shared with Epitalon
Cognitive, LongevitySPECULATIVE
155Piracetam
Original racetam-class nootropic (small molecule, pyrrolidone derivative)
CognitiveTIER 2 · Translational
156PNC-27
Synthetic 32-residue peptide combining an HDM-2 (MDM2) binding region from p53 with a membrane-residency leader; designed for tumour-selective membrane disruption
Cognitive, OtherTIER 3 · Preclinical
157PQQ
Pyrroloquinoline quinone (small molecule, redox cofactor); proposed mitochondrial biogenesis inducer
LongevityTIER 3 · Preclinical
158Pramlintide
Synthetic amylin analog (37-residue, 3 amino-acid substitutions for solubility)
MetabolicTIER 1 · Clinical
159Raloxifene
Selective estrogen receptor modulator (SERM); benzothiophene class
Sexual / hormonalTIER 1 · Clinical
160Rapamycin
Macrolide mTOR inhibitor (small molecule); endogenously produced by Streptomyces hygroscopicus
LongevityTIER 1 · Clinical
161Retatrutide
Triple agonist of GIP, GLP-1, and glucagon receptors
MetabolicTIER 2 · Translational
162Retatrutide + Cagrilintide (Blend)
Two-component blend — retatrutide (triple GLP-1/GIP/glucagon agonist) plus cagrilintide (long-acting amylin analog)
Blend, MetabolicTIER 2 · Translational
163Retatrutide + Tirzepatide (Blend)
Two-component blend — retatrutide (triple GLP-1/GIP/glucagon agonist) plus tirzepatide (dual GLP-1/GIP agonist)
Blend, MetabolicTIER 2 · Translational
164RG3 Snake Venom
Synthetic snake-venom mimetic peptide; topical cosmetic
CosmeticSPECULATIVE
165Secretin
Endogenous 27-residue gut peptide; secretin receptor (SCTR) agonist; foundational discovery hormone (Bayliss & Starling 1902)
Cognitive, MetabolicTIER 1 · Clinical
166Selank
Synthetic heptapeptide Thr-Lys-Pro-Arg-Pro-Gly-Pro (stabilized analog of tuftsin)
CognitiveTIER 3 · Preclinical
167Semaglutide
Long-acting GLP-1 receptor agonist
MetabolicTIER 1 · Clinical
168Semax
Synthetic heptapeptide Met-Glu-His-Phe-Pro-Gly-Pro (stabilized ACTH(4-10) fragment analog)
CognitiveTIER 3 · Preclinical
169Sermorelin
Synthetic GHRH(1-29)-NH2 — minimum bioactive fragment of endogenous GHRH
GH secretagogueTIER 1 · Clinical
170Setmelanotide
Synthetic melanocortin-4 receptor (MC4R) selective agonist; cyclic 8-residue peptide
MetabolicTIER 1 · Clinical
171Sigumir
Khavinson-tradition joint cartilage bioregulator (AED variant)
Longevity, HealingSPECULATIVE
172Sildenafil
Phosphodiesterase type 5 (PDE-5) inhibitor; pyrazolopyrimidinone class
Sexual / hormonalTIER 1 · Clinical
173Sincalide
Synthetic CCK-8 octapeptide; CCK-A and CCK-B receptor agonist
Cognitive, MetabolicTIER 1 · Clinical
174SLU-PP-332
Estrogen-related receptor (ERR) agonist (small molecule)
MetabolicTIER 3 · Preclinical
175SNAP-8
Synthetic acetylated octapeptide; INCI 'Acetyl Octapeptide-3'; SNARE complex / SNAP-25 mimic
CosmeticSPECULATIVE
176Somatropin
Recombinant 191-amino-acid human growth hormone
GH secretagogueTIER 1 · Clinical
177Spermidine
Endogenous polyamine; autophagy inducer (small molecule)
LongevityTIER 3 · Preclinical
178Splenopentin
Synthetic pentapeptide derived from splenin
ImmuneSPECULATIVE
179SR-9009
REV-ERB nuclear receptor agonist (small molecule)
MetabolicTIER 3 · Preclinical
180SS-31
Synthetic mitochondria-targeted tetrapeptide that binds cardiolipin in the inner mitochondrial membrane
CognitiveTIER 2 · Translational
181Substance P
Endogenous undecapeptide; tachykinin family; NK1 receptor agonist
CognitiveTIER 3 · Preclinical
182Survodutide
Dual GLP-1 / glucagon receptor agonist (Boehringer Ingelheim + Zealand Pharma)
MetabolicTIER 2 · Translational
183Syn-Ake
Synthetic tripeptide; INCI 'Tripeptide-3'; beta-Ala-Pro-Dab-NHBn benzylamide; snake-venom (waglerin) mimetic
CosmeticSPECULATIVE
184Tadalafil
Phosphodiesterase type 5 (PDE-5) inhibitor; β-carboline class
Sexual / hormonalTIER 1 · Clinical
185Tamoxifen
Selective estrogen receptor modulator (SERM); triphenylethylene class
Sexual / hormonalTIER 1 · Clinical
186TB-500
Naturally occurring 43-amino-acid peptide (Tβ4); TB-500 often used commercially as a synonym though technically refers to a synthetic fragment
HealingTIER 2 · Translational
187Teduglutide
Recombinant analog of GLP-2; selective GLP-2 receptor agonist
MetabolicTIER 1 · Clinical
188Teriparatide
Recombinant human parathyroid hormone amino acids 1-34
OtherTIER 1 · Clinical
189Tesamorelin
Stabilized human growth hormone-releasing hormone (1-44) analog
GH secretagogueTIER 1 · Clinical
190Tesamorelin + Ipamorelin (Blend)
Two-component vendor blend — tesamorelin (long-acting GHRH analog) plus ipamorelin (selective GHS-R1a agonist hexapeptide)
Blend, GH-stackSPECULATIVE
191Tesofensine
Triple monoamine reuptake inhibitor (noradrenaline, dopamine, serotonin)
MetabolicTIER 2 · Translational
192Testagen
Khavinson-tradition tetrapeptide (Lys-Glu-Asp-Gly); proposed thymus / immune bioregulator
Longevity, ImmuneSPECULATIVE
193Tetrahydrocurcumin-Peptide
Tetrahydrocurcumin-peptide hybrid conjugate (cosmetic)
CosmeticSPECULATIVE
194Tetrapeptide-21
Synthetic tetrapeptide; INCI 'Tetrapeptide-21'; photoaging-focused cosmetic peptide
CosmeticSPECULATIVE
195Thymalin
Fractionated peptide complex (multiple low-MW thymic peptides; not a defined single molecule)
ImmuneTIER 3 · Preclinical
196Thymogen
Synthetic dipeptide — L-glutamyl-L-tryptophan
ImmuneTIER 3 · Preclinical
197Thymosin Alpha-1
28-amino-acid peptide derived from prothymosin alpha
HealingTIER 2 · Translational
198Thymosin Beta-4 (TB-4)
Endogenous 43-residue actin-sequestering peptide; expressed by gene TMSB4X
HealingTIER 2 · Translational
199Thymulin
9-amino-acid thymic peptide; biologically active only when bound to zinc
HealingTIER 3 · Preclinical
200Tirzepatide
Dual GIP / GLP-1 receptor agonist
MetabolicTIER 1 · Clinical
201Tuftsin
Endogenous tetrapeptide — produced by leukokininase cleavage of IgG Fc; synthesised commercially
ImmuneTIER 3 · Preclinical
202Urolithin A
Gut microbial metabolite of ellagitannins; mitophagy inducer (small molecule)
LongevityTIER 2 · Translational
203Vasoactive Intestinal Peptide (VIP)
Vasoactive Intestinal Peptide; 28-residue secretin-family peptide; VPAC1/VPAC2 receptor agonist
CognitiveTIER 3 · Preclinical
204VEGF (Vascular Endothelial Growth Factor, research)
Endogenous secreted glycoprotein growth factor; multiple isoforms (VEGF121, VEGF165, VEGF189, VEGF206 from alternative splicing)
HealingTIER 3 · Preclinical
205Ventfort
Khavinson-tradition vascular bioregulator (KED-class variant)
LongevitySPECULATIVE
206Vesugen
Khavinson-tradition tripeptide (Lys-Glu-Asp); proposed vascular endothelium bioregulator
LongevitySPECULATIVE
207Vilon
Khavinson-tradition dipeptide (Lys-Glu); proposed thymus / immunomodulating bioregulator
Longevity, ImmuneSPECULATIVE
208Zhenagen
Khavinson-tradition testicular / reproductive bioregulator
LongevitySPECULATIVE
209α-MSH (Alpha Melanocyte-Stimulating Hormone)
Endogenous tridecapeptide derived from POMC processing; native melanocortin receptor agonist
Sexual / hormonal, CosmeticTIER 3 · Preclinical

◉ Pass % / N columns populate as our blind-purchase assay program brings samples through the lab queue. Until then, the compound list is organized by evidence tier and category only.